Ibuprofen-Standard--生命科学试剂-MCE.pdf

Hotline:400-820-3792

Inhibitors•ScreeningLibraries•Proteins

www.MedChemE

Ibuprofen(Standard)

Cat.No.:HY-78131R

CASNo.:15687-27-1

分⼦式:C₁₃H₁₈O₂

分⼦量:206.28

作⽤靶点:COX;Apoptosis;Parasite

作⽤通路:Immunology/Inflammation;Apoptosis;Anti-infection

储存⽅式:Pleasestoretheproductundertherecommendedconditionsin

theCertificateofAnalysis.

BIOLOGICALACTIVITY

⽣物活性Ibuprofen(Standard)是Ibuprofen的分析标准品。本产品⽤于研究及分析应⽤。Ibuprofen((±)-Ibuprofen)

是⼀种⼝服有效的COX-1选择性抑制剂，IC50值为13μM。Ibuprofen抑制细胞增殖、⾎管⽣成，并诱导细

胞凋亡(apoptosis)。Ibuprofen是⼀种⾮甾体抗炎试剂和⼀氧化氮(NO)供体。Ibuprofen可⽤于疼痛、肿胀、

炎症、感染、免疫学、癌症的研究。

IC50TargetIC50:13μM(COX-1),370μM(COX-2)

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